Argipressin (Arg8-vasopressin) binds to the V1, V2, V3-vascular arginine vasopressin receptor, with a Kd value of 1.31 nM in A7r5 rat aortic smooth muscle cells for V1.
体外研究
Argipressin binds to the vascular arginine vasopressin receptor, V1, with a Kd value of 1.31 nM in A7r5 rat aortic smooth muscle cells. It also stimulates the intracellular release of calcium in A7r5 cells (EC50=5 nM). AVP-induced [Ca]i signals and immunized activity against S-100 in DRG cell culture. The minimum effective concentrations of Argipressin causing [Ca]i responses are 100 pM in non-neuronal cells in DRG culture.
分子式
C46H65N15O12S2
分子量
1084.23
CAS号
113-79-1
中文名称
精氨加压素
运输条件
Room temperature in continental US; may vary elsewhere.