UNC 9994 hydrochloride
目录号 : KA1363
CAS No. : 2108826-33-9
纯度 : 98%
Unique, β-arrestin-biased functionally selective dopamine D2 receptor (D2R) agonist (Ki value 30 nM; EC50 value 50 nM in β-arrestin-2 recruitment assay) that exhibits antipsychotic activity in vivo. UNC9994 markedly inhibited PCP-induced hyperlocomotion in wild-type mice, which effect was completely abolished in β-arrestin-2 knockout mice.
Other Forms of Rapamycin:
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分子式 |
C21H22Cl2N2Os.HCl
|
分子量 |
457.84
|
CAS号 |
2108826-33-9
|