AY 77 is a potent PAR2 biased agonist. AY 77 exhibits bias for Ca2+over ERK1/2 signaling(EC50values are40 nM for Ca2+release versus 2 μM for ERK1/2 phosphorylation). Shows selectivity for PAR2 over PAR1. Promotes migration of human breast cancer cellsin vitro.
AY 77 is a potent PAR2 biased agonist. AY 77 exhibits bias for Ca2+over ERK1/2 signaling(EC50values are40 nM for Ca2+release versus 2 μM for ERK1/2 phosphorylation). Shows selectivity for PAR2 over PAR1. Promotes migration of human breast cancer cellsin vitro.
分子式
C21H32N4O4
分子量
404.511
CAS号
1835734-92-3
中文名称
AY77
运输条件
Room temperature in continental US; may vary elsewhere.