AY 77
目录号 : KE7657
CAS No. : 1835734-92-3
纯度 : ≥95%
AY 77 is a potent PAR2 biased agonist. AY 77 exhibits bias for Ca2+over ERK1/2 signaling(EC50values are40 nM for Ca2+release versus 2 μM for ERK1/2 phosphorylation). Shows selectivity for PAR2 over PAR1. Promotes migration of human breast cancer cellsin vitro.
Other Forms of Rapamycin:
KKL Med 的所有产品和服务仅用于科学研究,不能被用于人体,兽医,我们也不向个人提供产品和服务。
KKL 顾客使用本产品发表的 0 篇科研文献
暂无科研文献
生物活性 |
AY 77 is a potent PAR2 biased agonist. AY 77 exhibits bias for Ca2+over ERK1/2 signaling(EC50values are40 nM for Ca2+release versus 2 μM for ERK1/2 phosphorylation). Shows selectivity for PAR2 over PAR1. Promotes migration of human breast cancer cellsin vitro.
|
分子式 |
C21H32N4O4
|
分子量 |
404.511
|
CAS号 |
1835734-92-3
|
中文名称 |
AY77
|
运输条件 |
Room temperature in continental US; may vary elsewhere.
|
储存方式 |
Store at -20˚C
|