| 生物活性 |
CPI-455 is a specific KDM5 inhibitor withIC50 value of 10 ± 1 nM for full-length KDM5A in enzymatic assays, elevating global levels of H3K4 trimethylation (H3K4me3) and decreased the number of DTPs in multiple cancer cell line models treated with targeted agents or standard chemotherapy.
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| 分子式 |
C16H15ClN4O
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| 分子量 |
314.77
|
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| CAS号 |
2095432-28-1
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| 中文名称 |
CPI-455 hydrochloride
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| 运输条件 |
Room temperature in continental US; may vary elsewhere.
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| 储存方式 |
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纯度： ≥95%
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