Abemaciclib metabolite M2 (LSN2839567) is a metabolite of Abemaciclib, acts as a potent CDK4 and CDK6 inhibitor, with IC50s in the range of 1-3 nM. Anti-cancer activity.
IC50&Target
CDK4
1-3 nM (IC50)
CDK6
1-3 nM (IC50)
分子式
C25H28F2N8
分子量
478.54
CAS号
1231930-57-6
运输条件
Room temperature in continental US; may vary elsewhere.