Flumatinib mesylate (HHGV678 mesylate) is an orally available, selective inhibitor of Bcr-Abl. Flumatinib mesylate inhibits c-Abl, PDGFRβ and c-Kit with IC50s of 1.2 nM, 307.6 nM and 665.5 nM, respectively.
分子式
C29H29N8OF3.CH4O3S
分子量
658.69
CAS号
895519-91-2
中文名称
甲磺酸氟马替尼;甲磺酸氟马替尼/氟马替尼
运输条件
Room temperature in continental US; may vary elsewhere.