Devimistat (CPI-613) is a mitochondrial metabolism inhibitor. Devimistat is a lipoic acid antagonist that abrogates mitochondrial energy metabolism to induce apoptosis in various cancer cells.
IC50&Target
mitochondrial metabolism
体外研究
Devimistat induces apoptosis of GPM-2 gastric cancer cells. Devimistat targets the altered form of mitochondrial energy metabolism utilized by tumor cells. The change in mitochondrial enzyme activities and cellular redox status induced by devimistat leads to cell death, including apoptosis.
分子式
C22H28O2S2
分子量
388.59
CAS号
95809-78-2
运输条件
Room temperature in continental US; may vary elsewhere.