BSJ-03-123 is a PROTAC connected by ligands for Cereblon and CDK as a potent and novel CDK6-selective small-molecule degrader.
IC50&Target
CDK6
Cereblon
体外研究
BSJ-03-123 (BSJ) causes a pronounced anti-proliferative effect in CDK6-dependent AML cell lines by inducing a G1 cell-cycle arrest without a measurable increase in apoptosis.
分子式
C47H56N10O11
分子量
937.01
CAS号
2361493-16-3
运输条件
Room temperature in continental US; may vary elsewhere.