GSK467 is a cell penetrant and selective KDM5B (JARID1B or PLU1) inhibitor with a Ki of 10 nM, shows 180-fold selectivity for KDM4C and no measurable inhibitory effects toward KDM6 or other Jumonji family members.
IC50&Target
Ki: 10 nM (KDM5B)
分子式
C17H13N5O2
分子量
319.32
CAS号
1628332-52-4
运输条件
Room temperature in continental US; may vary elsewhere.