Aurora kinase inhibitor-2 is a selective and ATP-competitive Aurora kinase inhibitor with IC50s of 310 nM and 240 nM for Aurora A and Aurora B, respectively.
IC50&Target
Aurora A
310 nM (IC50)
Aurora B
240 nM (IC50)
体外研究
Aurora kinase inhibitor-2 (Compound 1) shows excellent levels of Aurora A enzyme inhibition and is also effective in an MCF7 cellular anti-proliferative assay (IC50 value of 1.25 µM).
分子式
C23H20N4O3
分子量
400.43
CAS号
331770-21-9
运输条件
Room temperature in continental US; may vary elsewhere.