[Ala17]-MCH, a MCH analogue , is a selective ligand for MCHR1 (Ki=0.16 nM) over MCHR2 (Ki=34 nM). [Eu chelate-labeled [Ala17]-MCH shows high affnity for MCHR1 (Kd=0.37 nM) while has little demonstrable binding affnity for MCHR2.
IC50&Target
Ki: 0.16 nM (MCHR1) Ki: 34 nM (MCHR2)
分子式
C97H155N29O26S4
分子量
2271.71
CAS号
359784-84-2
运输条件
Room temperature in continental US; may vary elsewhere.