Lonidamine (AF-1890), an antitumor agent, is a hexokinase, mitochondrial pyruvate carrier (Ki 2.5 μM in isolated rat liver mitochondria) and plasma membrane monocarboxylate transporters inhibitor, which also inhibits mitochondrial complex II.
IC50&Target
Ki: 2.5 μM (Mitochondrial pyruvate carrier)
分子式
C15H10Cl2N2O2
分子量
321.16
CAS号
50264-69-2
中文名称
氯尼达明;洛尼达酸;若丹明
运输条件
Room temperature in continental US; may vary elsewhere.