Bazedoxifene-d4 (acetate) is the deuterium labeled Bazedoxifene. Bazedoxifene (TSE-424) is an oral, BBB-penetrant nonsteroidal selective estrogen receptor modulator (SERM), with IC50s of 23 nM and 99 nM for ERα and ERβ, respectively. Bazedoxifene can be used for the research of osteoporosis. Bazedoxifene also acts as an inhibitor of IL-6/GP130 protein-protein interactions and can be used for the research of pancreatic cancer.
分子式
C32H34D4N2O5
分子量
534.68
CAS号
1795027-71-2
中文名称
[2H4]-苯多昔芬醋酸盐
运输条件
Room temperature in continental US; may vary elsewhere.