653-47 是一种增强剂，能显著增强 666-15 的 cAMP 反应元件结合蛋白 (CREB) 抑制活性。653-47 也是一种很弱的抑制剂，其 IC50 为 26.3 μM。
| 生物活性 |
653-47, a potentiator, significantly potentiates the cAMP-response element binding protein (CREB) inhibitory activity of 666-15. 653-47 is also a very weak CREB inhibitor with IC50 of 26.3 μM. |
|---|---|
| 体外研究 |
653-47 (5-10 μM) synergistically inhibits CREB-mediated gene transcription with 666-15. |
| 分子式 |
C20H19ClN2O3
|
| 分子量 |
370.83
|
| CAS号 |
1224678-75-4
|
| 运输条件 |
Room temperature in continental US; may vary elsewhere. |
| 储存方式 |
Please store the product under the recommended conditions in the Certificate of Analysis. |
关注我们
获得KKL MED 最新资讯
客服小K 
客服小K
Data Sheet