Almorexant (ACT 078573) is a potent and competitive dual orexin 1 receptor (OX1)/orexin 2 receptor (OX2) antagonist with Ki values of 1.3 and 0.17 nM, respectively.
IC50&Target
IC50: 1.3/0.7 nM(OX1/OX2 Receptor)
分子式
C29H31F3N2O3
分子量
512.56
CAS号
871224-64-5
运输条件
Room temperature in continental US; may vary elsewhere.