Fosaprepitant dimeglumine - CAS:265121-04-8

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Fosaprepitant dimeglumine (Synonyms:福沙吡坦二甲葡胺; MK-0517; L785298)

目录号 : KM8948 CAS No. : 265121-04-8 纯度 : 98%

Data Sheet 产品使用指南

Fosaprepitant dimeglumine (MK-0517) 是 Aprepitant 的前药。Fosaprepitant dimeglumine 是一种神经激肽-1 受体 (neurokinin-1 receptor) 拮抗剂，被开发用于预防化疗引起的恶心呕吐 (CINV)。

规格	价格	是否有货
5mg		In-stock
10mg		In-stock
50mg		In-stock
100mg		In-stock
200mg	询价	In-stock
500mg	询价	In-stock

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生物活性

Fosaprepitant dimeglumine (MK-0517) is a prodrug of Aprepitant . Fosaprepitant dimeglumine is a neurokinin-1 receptor antagonist, which is development for the prevention of chemotherapy-induced nausea and vomiting (CINV).

体内研究

Fosaprepitant dimeglumine (30 mg/kg; i.p.; daily; for 7 days) attenuates tolerance to morphine and increases the antinociceptive effect in in rats.

Animal Model:	Sprague-Dawley rats
Dosage:	30 mg/kg
Administration:	Intraperitoneal injection, daily, for 7 days
Result:	Increased the antinociceptive effect of morphine compared to control group.

分子式

C₃₇H₅₆F₇N₆O₁₆P

分子量

1004.83

CAS号

265121-04-8

中文名称

福沙吡坦二甲葡胺

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Powder	-20°C	3 years
	4°C	2 years

*该产品在溶液状态不稳定，建议您现用现配，即刻使用。

溶解性数据

In Vitro:

H₂O : 50 mg/mL (49.76 mM; Need ultrasonic)

配制储备液

浓度溶剂体积质量	1 mg	5 mg	10 mg

1 mM	0.9952 mL	4.9760 mL	9.9519 mL
5 mM	0.1990 mL	0.9952 mL	1.9904 mL
10 mM	0.0995 mL	0.4976 mL	0.9952 mL

请根据产品在不同溶剂中的溶解度，选择合适的溶剂配制储备液；该产品在溶液状态不稳定，建议您现用现配，即刻使用。

临床试验

科研文献

纯度： 98%

Data Sheet

产品使用指南

摩尔计算器
稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量

浓度

体积

分子量*

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
This equation is commonly abbreviated as: C1V1 = C2V2

浓度

体积

浓度

体积

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Other Forms of Rapamycin:

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The molarity calculator equation

The dilution calculator equation