AS2717638 is an oral active and selective lysophosphatidic acid receptor 5 (LPA5) antagonist, with an IC50 of 38 nM for hLPA5. AS2717638 also significantly improves PGE2-, PGF2α-, and AMPA-induced allodynia.
IC50&Target
IC50: 38 nM (hLPA5).
分子式
C25H25N3O5
分子量
447.48
CAS号
2148339-28-8
运输条件
Room temperature in continental US; may vary elsewhere.