Ulipristal Acetate-d6 - CAS:1621894-64-1

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Ulipristal Acetate-d6 (Synonyms:醋酸乌利司他-d6)

目录号 : KCM11809 CAS No. : 1621894-64-1 纯度 : 98%

Data Sheet 产品使用指南

Ulipristal acetate-d is intended for use as an internal standard for the quantification of ulipristal acetate by GC- or LC-MS. Ulipristal acetate is a selective progesterone receptor modulator (SPRM) that binds to the human progesterone receptors PR-A and PR-B (ECs = 8.5 and 7.7 nM, respectively), rabbit uterine PR (EC = 13.6 nM), and rabbit thymic glucocorticoid receptor (GR; EC = 15.4 nM). It is selective for human progesterone receptors over the human estrogen receptor (ER; EC = >10,000 nM). It inhibits growth of IGROV-1 and SK-OV-3 human ovarian cancer cells (ICs = 15.5 and 31.5 μM, respectively) even after resistance to combined cisplatin and paclitaxel treatment has developed. Ulipristal acetate reverses the proliferative effect of progesterone on patient-derived germline mutant BRCA1 breast tissue xenografts in ovariectomized athymic mice. Ulipristal acetate (40 mg/kg, i.p.) administered to female mice within 6 hours of human chorionic gonadotropin (hCG) treatment inhibits ovulation. Formulations containing ulipristal acetate have been used as emergency contraceptives and to treat uterine fibroids.

规格	价格	是否有货	数量
500μg		In-stock
1mg		In-stock

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Other Forms of Rapamycin:

XIE62-1004-A In-stock
SI-W052 In-stock
Biotin-16-UTP In-stock
Triphenyl phosphate In-stock
Ulipristal acetate-d3 In-stock

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生物活性

Ulipristal acetate-d6 is deuterium labeled Ulipristal acetate. Ulipristal acetate (CDB-2914) is an orally active, selective progesterone receptor modulator (SPRM). Ulipristal acetate stimulates the autophagic response selectively in leiomyoma cells. Ulipristal acetate has the potential for benign gynecological conditions treatment, such as uterine myoma.

分子式

C₃₀H₃₁D₆NO₄

分子量

481.65548

CAS号

1621894-64-1

中文名称

醋酸乌利司他-d6

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Powder	-20°C	3 years
	4°C	2 years
In solvent	-80°C	6 months
	-20°C	1 month

纯度： 98%

Data Sheet

产品使用指南

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The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
This equation is commonly abbreviated as: C1V1 = C2V2

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动物实验计算换算器

第一步：请输入基本实验信息（考虑到实验过程中的损耗，建议多配一只动物的药量）

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第二步：请输入动物体内配方组成（配方适用于不溶于水的药物；不同批次药物配方比例不同，请联系客服为您提供正确的澄清溶液配方）

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% Tween 80

% ddH₂O

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计算结果:

工作液浓度： mg/ml；

DMSO母液配制方法： mg 药物溶于 μL DMSO溶液（母液浓度 mg/mL，注：如该浓度超过该批次药物DMSO溶解度，请先联系客服）；

体内配方配制方法：取 μL DMSO母液，加入 μL PEG300，混匀澄清后加入μL Tween 80，混匀澄清后加入 μL ddH₂O，混匀澄清。

配置后的溶液总体积：

注意：1. 首先保证母液是澄清的；
2. 一定要按照顺序依次将溶剂加入，进行下一步操作之前必须保证上一步操作得到的是澄清的溶液，可采用涡旋、超声或水浴加热等物理方法助溶。

Other Forms of Rapamycin:

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The molarity calculator equation

The dilution calculator equation

动物实验计算换算器