(+)-ZK 216348
(Synonyms:(+)-ZK 216348)
目录号 : KA1526
CAS No. : 669073-68-1
纯度 : 98%
Selective nonsteroidal glucocorticoid receptor (GR) agonist for the treatment of experimental colitis with IC50 values of 20, 20, and 80 nM for GR, Progesterone (PR) and Mineralocorticoid (MR) receptors respectively. (+)-ZK 216348 shows antiinflammatory activity comparable to prednisolone for both systemic and topical application, with a significant dissociation between transrepression and transactivation of antiinflammatory effects both in vitro and in vivo.(+)-ZK 216348 showed no negative effects on intestinal epithelial migration or proliferation. (-)-ZK 216348 is completely inactive (IC50 >1000 nM for GR, PR, and MR.
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| 分子式 |
C24H23F3N2O5
|
| 分子量 |
476.45
|
| CAS号 |
669073-68-1
|
| 中文名称 |
(+)-ZK 216348
|
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