SAFit1 is a FK506 binding protein 51 (FKBP51)-specific inhibitor with a Ki of 4±0.3 nM.
IC50&Target
Ki: 4±0.3 nM (FKBP51), >50000 nM (FKBP52)
体外研究
SAFit1 (1-1000 nM) potently stimulates neurite outgrowth in two neuronal cell lines (N2a and SH-SY5Y) as well as in primary hippocampal neurons. SAFit1 is active over a wide concentration range.
分子式
C42H53NO11
分子量
747.87
CAS号
1643125-32-9
运输条件
Room temperature in continental US; may vary elsewhere.