GSK-843 (GSK'843) is a receptor-interacting protein kinase 3 (RIP3 or RIPK3) inhibitor, which binds RIP3 kinase domain with an IC50 of 8.6 nM, and inhibits kinase activity with an IC50 of 6.5 nM.
IC50&Target
IC50: 6.5 nM (RIP3)
分子式
C19H15N5S2
分子量
377.49
CAS号
1601496-05-2
运输条件
Room temperature in continental US; may vary elsewhere.