Arimoclomol maleate (BRX-220) is a co-inducer of heat shock proteins (HSP). Arimoclomol protects motor neurons by enhancing Hsp expression, thus directly affecting protein aggregation and clearance of misfolded assemblies via the proteasome-ubiquitin system.
体内研究
Arimoclomol (BRX-220; 20 mg/kg; orally administered for 5 d) has a protective effect against cholecystokinin-octapeptide (CCK)-induced acute pancreatitis.
Animal Model:
Male Wistar rats weighing 240 to 270 g
Dosage:
20 mg/kg
Administration:
Administered intragastrically, for 5 days
Result:
Had a protective effect against CCK-induced acute pancreatitis.
分子式
C14H20N3O3Cl.C4H4O4
分子量
429.85
CAS号
289893-26-1
运输条件
Room temperature in continental US; may vary elsewhere.