Naloxone HCl
(Synonyms:盐酸纳洛酮;17-烯丙基-4,5a-环氧基-3,14-二羟基吗啡喃-6-酮盐酸盐;17-烯丙基-4,5α-环氧-3,14-二羟基吗啡烷-6-酮;盐酸纳络酮;纳洛酮盐酸盐;盐酸纳诺酮;(-)-纳洛酮 盐酸盐;N-(1-(苯基乙酰基)-L-脯氨酰)甘氨酸乙酯;盐酸纳洛酮Naloxone hydrochloride)
目录号 : KF1065
CAS No. : 357-08-4
纯度 : 98%
Naloxone (357-08-4) is a pan-opioid receptor antagonist, Ki=3.7, 9.2 and 33 nM for m, k and d opioid receptors respectively. In clinical use in opiate abuse and overdose rescue. Blocks opiate- promoted wound healing. Attenuates the pruritic response to rimonabant in a rat model.
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| 分子式 |
C19H21NO4 &AmP;BUL;HCl
|
| 分子量 |
363.84
|
| CAS号 |
357-08-4
|
| 中文名称 |
盐酸纳洛酮
|
| 储存方式 |
| Powder |
-20°C |
3 years |
| |
4°C |
2 years |
| In solvent |
-80°C |
6 months |
| |
-20°C |
1 month |
|