Naloxone methiodide is a peripherally restricted, nonselective, and competitive opioid receptor antagonist. Naloxone methiodide does not penetrate the blood-brain barrier.
体内研究
Naloxone‐methiodide (10 mg/mL; 200 μL; i.p.), induces abdominal hypersensitivity in IL-10 mice with colitis.
Animal Model:
Ten- to twelve-week-old IL-10 gene-deficient male (IL-10−/−) mice on C57BL/6 genetic background
Dosage:
10 mg/mL; 200 μL
Administration:
Intraperitoneally
Result:
In piroxicam-treated IL-10 mice induced abdominal pain.
分子式
C20H24NO4+.I-
分子量
469.31
CAS号
93302-47-7
运输条件
Room temperature in continental US; may vary elsewhere.