PROTAC BET-binding moiety 1 is a key intermediate for the synthesis of high-affinity BET inhibitors.
体外研究
The bromodomain and extra-terminal (BET) family proteins, consisting of BRD2, BRD3, BRD4, and testis-specific BRDT members, are epigenetic "readers" and play a key role in the regulation of gene transcription. BET proteins are considered to be attractive therapeutic targets for cancer and other human diseases.
分子式
C25H25N7O4
分子量
487.51
CAS号
2093387-77-8
运输条件
Room temperature in continental US; may vary elsewhere.