| 生物活性 |
THIP-d4 (Gaboxadol-d4) is the deuterium labeled THIP . THIP (Gaboxadol) is a selective extrasynaptic GABAA receptors (eGABARs) agonist (with blood-brain barrier permeability), shows an EC50 value of 13 μM for δ-GABAAR. THIP induces strong tense GABAA-mediated currents in layer 2/3 neurons, but shows on effect on miniature IPSCs. THIP can be used in studies of sleep disorders.
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| 分子式 |
C6H4D4N2O2
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| 分子量 |
144.16
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| CAS号 |
2748778-97-2
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| 运输条件 |
Room temperature in continental US; may vary elsewhere.
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| 储存方式 |
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