Rac-Nedisertib
目录号 : KG10920
CAS No. : 1637542-34-7
纯度 : 98%
Rac-Nedisertib (Rac-M3814) is a racemate of Nedisertib, a potent DNA-PK inhibitor, with an IC50 of <3 nM. DNA-PK|<3 nM (IC50)
Rac-Nedisertib (Compound 137) potently inhibits DNA-PK, with an IC50 of <3 nM for DNA-PK, 0.5-5 μM for cellular pDNA-PK and 15-25 μM for KV11.1 (hERG, human ether a-go-go related gene) )..
Other Forms of Rapamycin:
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分子式 |
C24H21ClFN5O3
|
分子量 |
481.91
|
CAS号 |
1637542-34-7
|
中文名称 |
(Rac)-Nedisertib | (Rac)-M3814 | DNA-PK
|
储存方式 |
Store at -20°C
|