CKI-7 (hydrochloride)
(Synonyms:CKI-7盐酸盐;N-(2-氨基乙基)-5-氯异喹啉-8-磺酰胺双盐酸盐;洛米茶碱)
目录号 : KCM10513
CAS No. : 1177141-67-1
纯度 : ≥98%
CKI-7 is an inhibitor of casein kinase 1 (CK1; K = 8.5 μM). It is selective for CK1 over CK2, PKC, CaM kinase II (CaMKII), and cyclic AMP-dependent protein kinase (ICs = 90, >1,000, 195, and 550 μM, respectively). CKI-7 inhibits phosphorylation of a peptide substrate by Leishmania CK1.2 by 50% when used at a concentration of 10 μM.
Other Forms of Rapamycin:
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分子式 |
C11H12ClN3O2S.2HCl
|
分子量 |
285.7507
|
CAS号 |
1177141-67-1
|
中文名称 |
洛米茶碱
|
储存方式 |
Powder |
-20°C |
3 years |
|
4°C |
2 years |
In solvent |
-80°C |
6 months |
|
-20°C |
1 month |
|