Foropafant (SR27417) 是一种高效、竞争性、选择性、可口服的血小板激活因子 (PAF) 受体拮抗剂，抑制 [3H]PAF 与其受体结合，Ki 值为 57 pM，比未被标记的 PAF 低至少 5 倍。Foropafant (SR27417) 有效抑制 PAF 诱导的兔和人血小板聚集。
| 生物活性 |
Foropafant (SR27417) highly potent, competitive, selective and orally active antagonist of platelet-activating factor (PAF) receptor, with a Ki value of 57 pM for [H]PAF binding, at least 5-fold lower than that of unlabeled PAF itself. Foropafant potently inhibits PAF-induced aggregation of rabbit and human platelets. |
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| 分子式 |
C28H40N4S
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| 分子量 |
464.72
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| CAS号 |
136468-36-5
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| 中文名称 |
福罗帕泛
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| 运输条件 |
Room temperature in continental US; may vary elsewhere. |
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| 储存方式 |
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纯度： 98%
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