Scyliorhinin II 是一种选择性的神经激肽-3 (neurokinin-3 tachykinin) 受体激动剂，对大鼠脑皮层的 neurokinin-3 受体的 Ki 值为 2.5 nM。
| 生物活性 |
Scyliorhinin II is a selective neurokinin-3 receptor agonist, with a Ki of 2.5 nM for neurokinin-3 receptor in rat cerebral cortex. |
|---|---|
| 体外研究 |
Scyliorhinin II is a neurokinin-3 selective tachykinin receptor, with a Ki of 2.5 nM for neurokinin-3 (NK-3) receptor in rat cerebral cortex. Scyliorhinin II has little effect on NK-1 and NK-2 receptors, with Ki (NK-1 receptor)/Ki (NK-3 receptor) and Ki (NK-2 receptor)/Ki (NK-3 receptor) of 176 and 200. |
| 体内研究 |
Scyliorhinin II produces potent, dose-related reciprocal hindlimb scratching about equipotently with an ED50 of 0.08 nmol via intracerebroventricularly (i.c.v.) administration in mice.
|
| 分子式 |
C77H119N21O26S3
|
| 分子量 |
1851.09
|
| CAS号 |
112748-19-3
|
| 运输条件 |
Room temperature in continental US; may vary elsewhere. |
| 储存方式 |
Please store the product under the recommended conditions in the Certificate of Analysis. |
关注我们
获得KKL MED 最新资讯
客服小K 
客服小K
Data Sheet