Mesembrine-d3 是 Mesembrine 的氘代物。Mesembrine ((+)-Mesembrine) 一种主要的生物碱，具有芳基八氢吲哚骨架。Mesembrine 是一种 5-HT 转运蛋白抑制剂，Ki 为 1.4 nM。Mesembrine 还抑制磷酸二酯酶 4B (PDE4B)，IC50 为 7.8 μM。
| 生物活性 |
Mesembrine-d3 ((+)-Mesembrine-d3) is the deuterium labeled Mesembrine. Mesembrine ((+)-Mesembrine) a main alkaloid that features an aryloctahydroindole skeleton. Mesembrine is a 5-HT transporter inhibitor with a Ki of 1.4 nM. Mesembrine also inhibits phosphodiesterase 4B (PDE4B) with an IC50 of 7.8 μM. |
|---|---|
| 体外研究 |
Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs. |
| 分子量 |
292.39
|
| CAS号 |
1346600-05-2
|
| 运输条件 |
Room temperature in continental US; may vary elsewhere. |
| 储存方式 |
Please store the product under the recommended conditions in the Certificate of Analysis. |
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